Levocetirizine Dihydrochloride was prepared from benzoyl chloride by acidylation, hydrogenation, cyclization with an overall yield of 8.05 %.

  • 以苯甲酰氯为原料,经酰化, 还原, 环合等反应合成左旋西替利嗪盐酸盐,反应总收率为8.05%.

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